I-Antibiotic yeMithi yeZilwanyana ekumgangatho ophezulu iFlorfenicol CAS 73231-34-2
I-Florfenicol sisibulali-ntsholongwane esisetyenziswa kakhulu kwizilwanyana esine-spectrum ebanzi ye-antibacterial, isiphumo esinamandla se-antibacterial, i-low minimum inhibitory concentration (MIC), ukhuseleko oluphezulu, ayinatyhefu, kwaye ayinantsalela. Ayinabungozi obunokubangela i-aplastic anemia kwaye ifanelekile kwiifama ezinkulu zokuzalela. Isetyenziswa kakhulu ukunyanga izifo zokuphefumla zenkomo ezibangelwa yi-Pasteurella kunye ne-Haemophilus bacteria. Inefuthe elihle lokunyanga ukubola kweenyawo zenkomo okubangelwa yi-Clostridium. Ikwasetyenziswa kwizifo ezosulelayo ezibangelwa yi-bacteria ebuthathaka kwiihagu nakwiinkukhu, kunye nezifo ze-bacteria kwiintlanzi.
Isalathisi
1. Imfuyo: yokuthintela nokunyanga isifo sesifuba sehagu, i-pleuropneumonia eyosulelayo, i-atrophic rhinitis, isifo semiphunga yehagu, isifo se-streptococcal esibangelwa kubunzima bokuphefumla, ukunyuka kobushushu, ukukhwehlela, ukukrwitshwa, ukuncipha kokutya, ukuphelelwa ngamandla, njl.njl., inefuthe elinamandla kwi-E. coli kunye nezinye izizathu zesisu sehagu esityheli nesimhlophe, i-enteritis, isisu segazi, isifo sokudumba njalo njalo.
2. Iinkukhu: ukuthintela nokunyanga iinkukhu ezibangelwa yi-E. coli, iSalmonella, iPasteurella kunye nezinye i-cholera, urhudo olumhlophe lwenkukhu, urhudo, urhudo olunganyangekiyo, isitulo esimhlophe esiluhlaza, isitulo esinamanzi, urhudo, i-intestinal mucous membrane punctiform okanye ukopha okusasazekayo, i-omphalitis, i-pericardium, isibindi, iintsholongwane, izifo zokuphefumla ezingapheliyo ze-mycoplasma, i-infectious rhinitis, i-turbidity yebhaluni, ukukhohlela, i-tracheal rales, njl.
3. Inefuthe elicacileyo kwi-serositis esulelayo, i-Escherichia coli kunye ne-Pseudomonas aeruginosa kumadada.
4.Kwiimveliso zasemanzini. Unyango lwesifo seentlanzi ezibangelwa yintsholongwane, zithathwa ngaphakathi.
Idosi: 10-15mg/kg (xa kuthelekiswa nobunzima bentlanzi), kabini ngemini (eli yeza liyavuselela, lahlulwe kabini), ngokubanzi iintsuku ezintathu kwikhosi yonyango. Iishrimp kunye neenkala zinamathumbu amafutshane. Phinda kabini idosi. Qaphela: Sebenzisa ngeentsuku ezinelanga.
I-Flufenicol iyahambelana nayo
1. Xa idibene ne-neomycin, i-doxycycline hydrochloride, i-colistin sulfate, i-loricin, njl.njl., isiphumo sokunyanga siyaphuculwa.
2. Xa idibene ne-ampicillin, i-cefradine, i-cephalexin, njl.njl., ukusebenza kwayo kuyancitshiswa.
3. Ukuhambelana ne-kanamycin, i-streptomycin, i-sulfonamides kunye ne-quinolones kwandisa ubuthi.
4. Ihambelana neVB12, inokuthintela i-erythropoiesis.
Isenzo sezonyango
Ingasasazwa kwiiseli zebhaktiriya ngokunyibilika kwamafutha, ikakhulu isebenza kwi-subunit yama-50s ye-ribosome yama-70s yebhaktiriya, ithintele i-transpeptidase, ithintele ukukhula kwe-peptidase, ithintele ukwakheka kwe-peptide chain, kwaye ngaloo ndlela ithintele ukwenziwa kweeproteni ukuze kufezekiswe iinjongo zokulwa ne-antibacterial. Le mveliso ine-spectrum ebanzi ye-antibacterial kwaye inefuthe elinamandla kwiibhaktiriya ze-Gram-positive kunye ne-Gram-negative kunye ne-mycoplasma. Le mveliso inokufunxwa ngokukhawuleza ngomlomo, isasazwa ngokubanzi, isiqingatha sobomi, uxinzelelo oluphezulu lweziyobisi egazini kunye nexesha elide lokugcinwa kweziyobisi egazini.










